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ESI Special Topic of:
"COX-2 Inhibitors," Published January 2005

•> Search Special Topics
COX-2 Inhibitors Menu

COX-2 Inhibitors

TOP PAPERS Top 20 papers overall

  
***Article 1
Special Topics Interview with Taketo, MM
Journal: CELL
Volume: 87
Page: 803-809
Year: 1996
Total Cites: 1115
Expected Cites: 248.92
Article Title: SUPPRESSION OF INTESTINAL POLYPOSIS IN APC(DELTA 716) KNOCKOUT MICE BY INHIBITION OF CYCLOOXYGENASE 2 (COX-2)
Authors: Oshima, M, Dinchuk, JE, Kargman, SL, Oshima, H, Hancock, B, Kwong, E, Trzaskos, JM, Evans, JF, Taketo, MM
Addresses: 
· BANYU TSUKUBA RES INST MERCK, TSUKUBA, IBARAKI 30033, JAPAN
· DUPONT MERCK PHARMACEUT CO, WILMINGTON, DE, USA
· MERCK & CO INC, POINTE CLAIRE, PQ H9R 4P8, CANADA
· UNIV TOKYO, FAC PHARMACEUT SCI, DEPT BIOMED GENET, BUNKYO KU, TOKYO 113, JAPAN

***Article 2
Journal: CELL
Volume: 93
Page: 705-716
Year: 1998
Total Cites: 885
Expected Cites: 188.33
Article Title: CYCLOOXYGENASE REGULATES ANGIOGENESIS INDUCED BY COLON CANCER CELLS
Authors: Tsujii, M, Kawano, S, Tsuji, S, Sawaoka, H, Hori, M, Dubois, RN
Addresses: 
· VANDERBILT UNIV, Med Ctr, Dept Med, VA Med Ctr, Nashville, TN, USA
· VANDERBILT UNIV, Med Ctr, Dept Med, VA Med Ctr, Nashville, TN, USA
· VANDERBILT UNIV, Med Ctr, Dept Cell Biol, Nashville, TN, USA
· OSAKA UNIV, Sch Med, Dept Med 1, Osaka 5650871, Japan

***Article 3
Journal: PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-PHYSICAL SCIENCES
Volume: 91
Page: 3228-3232
Year: 1994
Total Cites: 817
Expected Cites: 84.06
Article Title: SELECTIVE-INHIBITION OF INDUCIBLE CYCLOOXYGENASE-2 IN-VIVO IS ANTIINFLAMMATORY AND NONULCEROGENIC
Authors: Masferrer, JL, Zweifel, BS, Manning, PT, Hauser, SD, Leahy, KM, Smith, WG, Isakson, PC, Seibert, K
Addresses: 
· SEARLE & CO, SEARLE INFLAMMATORY DIS RES, 800 N LINDBERGH ST, ST LOUIS, MO, USA

***Article 4
Journal: ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY
Volume: 38
Page: 97-120
Year: 1998
Total Cites: 736
Expected Cites: 109.95
Article Title: CYCLOOXYGENASES 1 AND 2
Authors: Vane, JR, Bakhle, YS, Botting, RM
Addresses: 
· UNIV LONDON QUEEN MARY & WESTFIELD COLL, St Bartholomews & Royal London Sch Med & Dent, William Harvey Res Inst, Charterhouse Sq, London EC1M 6BQ, England
· UNIV LONDON QUEEN MARY & WESTFIELD COLL, St Bartholomews & Royal London Sch Med & Dent, William Harvey Res Inst, London EC1M 6BQ, England

***Article 5
Journal: NEW ENGLAND JOURNAL OF MEDICINE
Volume: 342
Page: 1946-1952
Year: 2000
Total Cites: 600
Expected Cites: 95.7
Article Title: THE EFFECT OF CELECOXIB, A CYCLOOXYGENASE-2 INHIBITOR, IN FAMILIAL ADENOMATOUS POLYPOSIS
Authors: Steinbach, G, Lynch, PM, Phillips, RKS, Wallace, MH, Hawk, E, Gordon, GB, Wakabayashi, N, Saunders, B, Shen, Y, Fujimura, T, Su, LK, Levin, B, Godio, L, Patterson, S, Rodriguez-bigas, MA, Jester, SL, King, KL, Schumacher, M, Abbruzzese, J, Dubois, RN, Hittelman, WN, Zimmerman, S, Sherman, JW, Kelloff, G
Addresses: 
· UNIV TEXAS, MD Anderson Canc Ctr, Div Canc Prevent, Box 203, Houston, TX, USA
· UNIV TEXAS, MD Anderson Canc Ctr, Div Canc Prevent, Houston, TX, USA
· ST MARKS HOSP, Imperial Canc Res Fund, London EC1V 2PS, England
· NCI, Bethesda, MD, USA
· SEARLE & CO, Skokie, IL, USA

***Article 6
Journal: CANCER RESEARCH
Volume: 58
Page: 409-412
Year: 1998
Total Cites: 466
Expected Cites: 46.66
Article Title: CHEMOPREVENTIVE ACTIVITY OF CELECOXIB, A SPECIFIC CYCLOOXYGENASE-2 INHIBITOR, AGAINST COLON CARCINOGENESIS
Authors: Kawamori, T, Rao, CV, Seibert, K, Reddy, BS
Addresses: 
· AMER HLTH FDN, Div Nutr Carcinogenesis, 1 Dana Rd, Valhalla, NY, USA
· AMER HLTH FDN, Div Nutr Carcinogenesis, Valhalla, NY, USA
· SEARLE & CO, St Louis, MO, USA

***Article 7
Journal: CANCER RESEARCH
Volume: 58
Page: 362-366
Year: 1998
Total Cites: 418
Expected Cites: 46.66
Article Title: MODULATION OF APOPTOSIS AND BCL-2 EXPRESSION BY PROSTAGLANDIN E-2 IN HUMAN COLON CANCER CELLS
Authors: Sheng, HM, Shao, JY, Morrow, JD, Beauchamp, RD, Dubois, RN
Addresses: 
· VANDERBILT UNIV, Med Ctr, Dept Med GI, MCN C-2104, Nashville, TN, USA
· VANDERBILT UNIV, Med Ctr, Dept Med, Nashville, TN, USA
· VANDERBILT UNIV, Med Ctr, Dept Cell Biol, Nashville, TN, USA
· VANDERBILT UNIV, Med Ctr, Dept Surg, Nashville, TN, USA
· VANDERBILT UNIV, Med Ctr, Ctr Mol Toxicol, Nashville, TN, USA
· VET ADM MED CTR, Nashville, TN, USA

***Article 8
Journal: JOURNAL OF MEDICINAL CHEMISTRY
Volume: 40
Page: 1347-1365
Year: 1997
Total Cites: 406
Expected Cites: 23.73
Article Title: SYNTHESIS AND BIOLOGICAL EVALUATION OF THE 1,5-DIARYLPYRAZOLE CLASS OF CYCLOOXYGENASE-2 INHIBITORS: IDENTIFICATION OF 4-[5-(4-METHYLPHENYL)-3-(TRIFLUOROMETHYL)-1H-PYRAZOL-1-YL]BENZENESULFONAMIDE (SC-58635, CELECOXIB)
Authors: Penning, TD, Talley, JJ, Bertenshaw, SR, Carter, JS, Collins, PW, Docter, S, Graneto, MJ, Lee, LF, Malecha, JW, Miyashiro, JM, Rogers, RS, Rogier, DJ, Yu, SS, Anderson, GD, Burton, EG, Cogburn, JN, Gregory, SA, Koboldt, CM, Perkins, WE, Seibert, K, Veenhuizen, AW, Zhang, YY, Isakson, PC
Addresses: 
· SEARLE & CO, DEPT CHEM, 4901 SEARLE PKWY, SKOKIE, IL, USA
· SEARLE & CO, DEPT INFLAMMATORY DIS RES, SKOKIE, IL, USA
· SEARLE & CO, DEPT MOL PHARMACOL, SKOKIE, IL, USA

***Article 9
Journal: NATURE
Volume: 384
Page: 644-648
Year: 1996
Total Cites: 405
Expected Cites: 172.76
Article Title: STRUCTURAL BASIS FOR SELECTIVE INHIBITION OF CYCLOOXYGENASE-2 BY ANTI-INFLAMMATORY AGENTS
Authors: Kurumbail, RG, Stevens, AM, Gierse, JK, Mcdonald, JJ, Stegeman, RA, Pak, JY, Gildehaus, D, Miyashiro, JM, Penning, TD, Seibert, K, Isakson, PC, Stallings, WC
Addresses: 
· SEARLE & CO, 700 CHESTERFIELD PKWY N, ST LOUIS, MO, USA
· SEARLE & CO, SKOKIE, IL, USA

***Article 10
Journal: LANCET
Volume: 353
Page: 307-314
Year: 1999
Total Cites: 383
Expected Cites: 36.61
Article Title: COX-2 INHIBITORS
Authors: Hawkey, CJ
Addresses: 
· UNIV NOTTINGHAM, Queens Med Ctr, Nottingham NG7 2UH, England
· UNIV NOTTINGHAM, Queens Med Ctr, Nottingham NG7 2UH, England

***Article 11
Journal: CANCER RESEARCH
Volume: 60
Page: 1306-1311
Year: 2000
Total Cites: 375
Expected Cites: 31.39
Article Title: ANTIANGIOGENIC AND ANTITUMOR ACTIVITIES OF CYCLOOXYGENASE-2 INHIBITORS
Authors: Masferrer, JL, Leahy, KM, Koki, AT, Zweifel, BS, Settle, SL, Woerner, BM, Edwards, DA, Flickinger, AG, Moore, RJ, Seibert, K
Addresses: 
· GD SEARLE MONSANTO CO, T3G, 800 N Lindbergh Blvd, St Louis, MO, USA
· GD SEARLE MONSANTO CO, St Louis, MO, USA

***Article 12
Journal: JAMA-JOURNAL OF THE AMERICAN MEDICAL ASSOCIATION
Volume: 282
Page: 1921-1928
Year: 1999
Total Cites: 358
Expected Cites: 77.04
Article Title: ANTI-INFLAMMATORY AND UPPER GASTROINTESTINAL EFFECTS OF CELECOXIB IN RHEUMATOID ARTHRITIS - A RANDOMIZED CONTROLLED TRIAL
Authors: Simon, LS, Weaver, AL, Graham, DY, Kivitz, AJ, Lipsky, PE, Hubbard, RC, Isakson, PC, Verburg, KM, Yu, SS, Zhao, WW, Geis, GS
Addresses: 
· HARVARD UNIV, Sch Med, Beth Israel Deaconess Med Ctr, Dept Med, Boston, MA, USA
· HARVARD UNIV, Sch Med, Beth Israel Deaconess Med Ctr, Dept Med, Boston, MA, USA
· ARTHRIT CTR NEBRASKA, Lincoln, NE, USA
· BAYLOR COLL MED, Vet Affairs Med Ctr, Dept Med, Houston, TX, USA
· Altoona Ctr Clin Res, Altoona, PA, USA
· UNIV TEXAS, SW Med Ctr, Div Rheumat Dis, Dallas, TX, USA
· SEARLE & CO, Dept Clin Res, Skokie, IL, USA
· SEARLE & CO, COX2 Technol, Skokie, IL, USA

***Article 13
Journal: JOURNAL OF CLINICAL INVESTIGATION
Volume: 99
Page: 2254-2259
Year: 1997
Total Cites: 351
Expected Cites: 67.89
Article Title: INHIBITION OF HUMAN COLON CANCER CELL GROWTH BY SELECTIVE INHIBITION OF CYCLOOXYGENASE-2
Authors: Sheng, HM, Shao, JY, Kirkland, SC, Isakson, P, Coffey, RJ, Morrow, J, Beauchamp, RD, Dubois, RN
Addresses: 
· VANDERBILT UNIV, MED CTR, DEPT MED, NASHVILLE, TN, USA
· VANDERBILT UNIV, MED CTR, DEPT SURG, NASHVILLE, TN, USA
· VANDERBILT UNIV, MED CTR, DEPT CELL BIOL, NASHVILLE, TN, USA
· VET ADM MED CTR, NASHVILLE, TN, USA
· SEARLE & CO, DEPT INFLAMMATORY DIS RES, ST LOUIS, MO, USA
· UNIV LONDON, ROYAL POSTGRAD MED SCH, IMPERIAL CANC RES FUND, HISTOPATHOL UNIT, LONDON W12 0NN, ENGLAND

***Article 14
Journal: NATURE MEDICINE
Volume: 5
Page: 698-701
Year: 1999
Total Cites: 338
Expected Cites: 113.02
Article Title: INDUCIBLE CYCLOOXYGENASE MAY HAVE ANTI-INFLAMMATORY PROPERTIES
Authors: Gilroy, DW, Colville-nash, PR, Willis, D, Chivers, J, Paul-clark, MJ, Willoughby, DA
Addresses: 
· ST BARTHOLOMEWS HOSP, Dept Expt Pathol, London EC1M 6BQ, England
· ST BARTHOLOMEWS HOSP, Dept Expt Pathol, London EC1M 6BQ, England

***Article 15
Journal: PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-PHYSICAL SCIENCES
Volume: 96
Page: 272-277
Year: 1999
Total Cites: 331
Expected Cites: 50.53
Article Title: SYSTEMIC BIOSYNTHESIS OF PROSTACYCLIN BY CYCLOOXYGENASE (COX)-2: THE HUMAN PHARMACOLOGY OF A SELECTIVE INHIBITOR OF COX-2
Authors: Mcadam, BF, Catella-lawson, F, Mardini, IA, Kapoor, S, Lawson, JA, Fitzgerald, GA
Addresses: 
· UNIV PENN, Stellar Chance Labs 905, Ctr Expt Therapeut, EUPENN Grp Investigators, Philadelphia, PA, USA
· UNIV PENN, Stellar Chance Labs 905, Ctr Expt Therapeut, EUPENN Grp Investigators, Philadelphia, PA, USA

***Article 16
Journal: JAMA-JOURNAL OF THE AMERICAN MEDICAL ASSOCIATION
Volume: 286
Page: 954-959
Year: 2001
Total Cites: 331
Expected Cites: 41.66
Article Title: RISK OF CARDIOVASCULAR EVENTS ASSOCIATED WITH SELECTIVE COX-2 INHIBITORS
Authors: Mukherjee, D, Nissen, SE, Topol, EJ
Addresses: 
· CLEVELAND CLIN FDN, Dept Cardiovasc Med, F 25, 9500 Euclid Ave, Cleveland, OH, USA
· CLEVELAND CLIN FDN, Dept Cardiovasc Med, Cleveland, OH, USA

***Article 17
Journal: ANNUAL REVIEW OF BIOCHEMISTRY
Volume: 69
Page: 145-182
Year: 2000
Total Cites: 330
Expected Cites: 119.48
Article Title: CYCLOOXYGENASES: STRUCTURAL, CELLULAR, AND MOLECULAR BIOLOGY
Authors: Smith, WL, Dewitt, DL, Garavito, RM
Addresses: 
· MICHIGAN STATE UNIV, Dept Biochem, E Lansing, MI, USA
· MICHIGAN STATE UNIV, Dept Biochem, E Lansing, MI, USA

***Article 18
Journal: NATURE MEDICINE
Volume: 5
Page: 1418-1423
Year: 1999
Total Cites: 303
Expected Cites: 113.02
Article Title: INHIBITION OF ANGIOGENESIS BY NONSTEROIDAL ANTI-INFLAMMATORY DRUGS: INSIGHT INTO MECHANISMS AND IMPLICATIONS FOR CANCER GROWTH AND ULCER HEALING
Authors: Jones, MK, Wang, HT, Peskar, BM, Levin, E, Itani, RM, Sarfeh, IJ, Tarnawski, AS
Addresses: 
· VET ADM MED CTR, Dept Med, 5901 E 7th St, Long Beach, CA, USA
· VET ADM MED CTR, Dept Med, Long Beach, CA, USA
· VET ADM MED CTR, Dept Surg, Long Beach, CA, USA
· UNIV CALIF IRVINE, Dept Med, Irvine, CA, USA
· UNIV CALIF IRVINE, Dept Surg, Irvine, CA, USA
· RUHR UNIV BOCHUM, Dept Expt Clin Med, D-44780 Bochum, Germany

***Article 19
Journal: ARTHRITIS AND RHEUMATISM
Volume: 41
Page: 1591-1602
Year: 1998
Total Cites: 284
Expected Cites: 30.96
Article Title: PRELIMINARY STUDY OF THE SAFETY AND EFFICACY OF SC-58635, A NOVEL CYCLOOXYGENASE 2 INHIBITOR - EFFICACY AND SAFETY IN TWO PLACEBO-CONTROLLED TRIALS IN OSTEOARTHRITIS AND RHEUMATOID ARTHRITIS, AND STUDIES OF GASTROINTESTINAL AND PLATELET EFFECTS
Authors: Simon, LS, Lanza, FL, Lipsky, PE, Hubbard, RC, Talwalker, S, Schwartz, BD, Isakson, PC, Geis, GS
Addresses: 
· HARVARD UNIV, Sch Med, Beth Israel Deaconess Med Ctr, Div Rheumatol & Metab Bone Dis, Boston, MA, USA
· HARVARD UNIV, Sch Med, Beth Israel Deaconess Med Ctr, Div Rheumatol & Metab Bone Dis, Boston, MA, USA
· HOUSTON INST CLIN RES, Houston, TX, USA
· UNIV TEXAS, SW Med Ctr, Dallas, TX, USA
· SEARLE & CO, Skokie, IL, USA

***Article 20
Journal: CANCER RESEARCH
Volume: 56
Page: 4566-4569
Year: 1996
Total Cites: 268
Expected Cites: 59.77
Article Title: EVALUATION OF CYCLOOXYGENASE-2 INHIBITOR FOR POTENTIAL CHEMOPREVENTIVE PROPERTIES IN COLON CARCINOGENESIS
Authors: Reddy, BS, Rao, CV, Seibert, K
Addresses: 
· AMER HLTH FDN, DIV NUTR CARCINOGENESIS, 1 DANA RD, VALHALLA, NY, USA
· SEARLE & CO, ST LOUIS, MO, USA

ESI Special Topic of:
"COX-2 Inhibitors," Published January 2005

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